反应条件
1: 87 percent / HMDS, TCS, C4F9SO3K / acetonitrile / 24 h / Heating 2: 95 percent / NH3 / methanol / 24 h / Ambient temperature 3: pyridine / 4 h / 0 °C 4: aq. NaOH / aq. ethanol / 135 h / Heating 5: 56 percent / H2 / 10percent Pd/C / methanol / 4 h / 2585.7 Torr / Ambient temperature View Scheme
参考文献
Lin, Tai-Shun; Zhu, Ju-Liang; Dutschman, Ginger E.; Cheng, Yung-Chi; Prusoff, William H.
Journal of Medicinal Chemistry, 1993 , vol. 36, # 3 p. 353 - 362
