反应条件
<b>Multi-step reaction with 4 steps<br /> </b>1: COCl<sub>2</sub>, DMF / CH<sub>2</sub>Cl<sub>2</sub> / Ambient temperature<br />2: CH<sub>2</sub>Cl<sub>2</sub> / Ambient temperature<br />3: SOCl<sub>2</sub> / CHCl<sub>3</sub> / Ambient temperature<br />4: 1) lithium diisopropylamide / 1) THF, -78 deg C, 2) up to room temp.<br /> <br />
参考文献
Hagen; Domagala Journal of Heterocyclic Chemistry, 1990 , vol. 27, # 6 p. 1609 - 1616