反应条件
1: tetrahydrothiophene 1,1-dioxide / 150 °C 2: 1.) NaH, DMSO / 1.) DMF, 2.) DMF View Scheme
参考文献
Hargrave, Karl D.; Proudfoot, John R.; Grozinger, Karl G.; Cullen, Ernest; Kapadia, Suresh R.; et al.
Journal of Medicinal Chemistry, 1991 , vol. 34, # 7 p. 2231 - 2241