反应条件
1: 1.) sodium hydride / 1.) DMF, 0 deg C, 30 min, 2.) DMF, 0 deg C, 30 min 2: 65 percent / AIBN, tri-n-butyltin hydride / toluene / 0.17 h / 90 °C 3: 88 percent / 80percent acetic acid / 0.58 h / 90 °C View Scheme
参考文献
Barchi, Joseph J.; Marquez, Victor E.; Driscoll, John S.; Ford, Harry; Mitsuya, Hiroaki; et al.
Journal of Medicinal Chemistry, 1991 , vol. 34, # 5 p. 1647 - 1655
