反应条件
1: 1.) pyridine / 1.) -10 deg C, overnight, 2.) RT, overnight 2: 80 percent / DBU / CH2Cl2 / 72 h / Ambient temperature 3: 42 percent / HF, AlF3 / dioxane / 1 h / 170 °C View Scheme
参考文献
Huang; Chen; Wang; Kim; Warshaw; Armstrong; Zhu; Chou; Watanabe; Matulic-Adamic; Su; Fox; Polsky; Baron; Gold; Hardy; Zuckerman
Journal of Medicinal Chemistry, 1991 , vol. 34, # 5 p. 1640 - 1646