1: 1) NaH / 1) RT, 0.5h, 2) RT
2: 44 percent / KF / dimethylsulfoxide / 2 h / 170 °C
View Scheme
参考文献
Jacobs, Robert T.; Bernstein, Peter R.; Cronk, Laura A.; Vacek, Edward P.; Newcomb, Lisa F.; et al.
Journal of Medicinal Chemistry, 1994 , vol. 37, # 9 p. 1282 - 1297