反应条件
1: piperidine / N,N-dimethyl-formamide / 1 h / 20 °C
2: N,O-bis-(trimethylsilyl)-acetamide; triethylamine / tetrahydrofuran / 10 h / 20 °C
View Scheme
参考文献
Wu, Wenting; Zhang, Zhihui; Liebeskind, Lanny S.
Journal of the American Chemical Society, 2011 , vol. 133, # 36 p. 14256 - 14259