1: With potassium phosphate; trifluoromethyl amino ketone; N-methyl-2-(methylamino)ethylamine; copper(l) iodide in N,N-dimethyl-formamide T=45°C; 2: With methanol in N,N-dimethyl-formamide T=45°C; Further stages.;
ammonia; bis-triphenylphosphine-palladium(II) chloride in tetrahydrofuran; water T=20°C; P=760 Torr; 30 h;
参考文献
Mohamed Ahmed, Mohamed S.; Sekiguchi, Akitoshi; Masui, Kentaro; Mori, Atsunori
Bulletin of the Chemical Society of Japan, 2005 , vol. 78, # 1 p. 160 - 168
