1: oxalyl chloride / CH2Cl2 / Heating 2: 0.37 g / Et2AlCl / CH2Cl2; hexane / 2 h / 20 °C View Scheme
参考文献
Eissenstat, Michael A.; Bell, Malcolm R.; D'Ambra, Thomas E.; Alexander, E. John; Daum, Sol J.; et al.
Journal of Medicinal Chemistry, 1995 , vol. 38, # 16 p. 3094 - 3105