反应条件
1: 80 percent / Et3N, DCC, DMAP / CH2Cl2 / 20 h / 25 °C 2: 100 percent / LiOH*H2O / tetrahydrofuran; methanol; H2O / 3 h / 25 °C View Scheme
参考文献
Andersen, Rikke; Nielsen, Carsten Uhd; Begtrup, Mikael; Jorgensen, Flemming Steen; Brodin, Birger; Frokjaer, Sven; Steffansen, Bente
European Journal of Pharmaceutical Sciences, 2006 , vol. 28, # 4 p. 325 - 335