反应条件
1: benzene / 26 h / Heating 2: tBuNH2, KN(TMS)2 3: 1.) BH3, 2.) NaOAc, H2O2 / 1.) THF, 23 deg C, 10 h, 2.) CH3OH, 23 deg C, 12 h 4: 85 percent / 6 N HCl / tetrahydrofuran / 12 h / 23 °C View Scheme
参考文献
Pearson; Lin
Tetrahedron Letters, 1990 , vol. 31, # 52 p. 7571 - 7574