反应条件
1: 81 percent / pyridine / 12 h / Ambient temperature 2: NaN3 / dimethylsulfoxide / 1 h / 180 °C 3: pyridine / 12 h / Ambient temperature 4: 58 percent / TMS-Tfl, bis(trimethylsilyl)thymine / acetonitrile / 3 h / Heating 5: 68 percent / ammonia / methanol / 48 h View Scheme
参考文献
Mikhailopulo; Poopeiko; Pricota; Sivets; Kvasyuk; Balzarini; De Clercq
Journal of Medicinal Chemistry, 1991 , vol. 34, # 7 p. 2195 - 2202