反应条件
1.1: N-ethyl-N,N-diisopropylamine / water; ethanol / 0.67 h / 60 °C 2.1: trimethylsilyl trifluoromethanesulfonate; N-ethyl-N,N-diisopropylamine / dichloromethane / 0.25 h / 20 °C / |Inert atmosphere 2.2: 0.33 h / |Inert atmosphere View Scheme
参考文献
Karoli, Tomislav; Becker, Bernd; Zuegg, Johannes; Moellmann, Ute; Ramu, Soumya; Huang, Johnny X.; Cooper, Matthew A.
Journal of Medicinal Chemistry, 2012 , vol. 55, # 17 p. 7940 - 7944
