反应条件
1: 3-bromo-2-hydroxypyridine With sodium hydride in DMF (N,N-dimethyl-formamide) T=20°C; 0.5 h; 2: benzyl bromide in DMF (N,N-dimethyl-formamide) T=20°C;
参考文献
Ding, Min; He, Feng; Hudyma, Thomas W.; Zheng, Xiaofan; Poss, Michael A.; Kadow, John F.; Beno, Brett R.; Rigat, Karen L.; Wang, Ying-Kai; Fridell, Robert A.; Lemm, Julie A.; Qiu, Dike; Liu, Mengping; Voss, Stacey; Pelosi, Lenore A.; Roberts, Susan B.; Gao, Min; Knipe, Jay; Gentles, Robert G.
Bioorganic and Medicinal Chemistry Letters, 2012 , vol. 22, # 8 p. 2866 - 2871