反应条件
1: 88 percent
2: 82 percent / N-Methylmorpholin, Ethylchlorformiat / CH2Cl2 / 16 h / -15 - 20 °C
3: 76 percent / Naphthalin-Na / 1,2-dimethoxy-ethane / 6 h / 0 - 20 °C
View Scheme
参考文献
Martens, Juergen; Scheunemann, Matthias
Tetrahedron Letters, 1991 , vol. 32, # 11 p. 1417 - 1418