1: 2-lt;2-lt;2-(aminoethoxy)ethoxygt;ethoxygt;acetic acid With potassium carbonate in water T=20°C; 0.25 h; 2: 1-[[(9H-fluoren-9-ylmethoxy)carbonyl]oxy]-2,5-pyrrolidinedione in water 24 h;
参考文献
Gomez, Francisco L. Guerra; Uehara, Tomoya; Rokugawa, Takemi; Higaki, Yusuke; Suzuki, Hiroyuki; Hanaoka, Hirofumi; Akizawa, Hiromichi; Arano, Yasushi
Bioconjugate Chemistry, 2012 , vol. 23, # 11 p. 2229 - 2238