1.1: NH2OH*HCl; Na2CO3 / ethanol; H2O / 1 h / 60 °C 2.1: N-chlorosuccinimide; pyridine / tetrahydrofuran / 0.5 h / 60 °C 2.2: triethylamine / tetrahydrofuran / 2 h / 50 °C View Scheme
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sodium cyanoborohydride in methanol T=20°C; Inert atmosphere;
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