反应条件
1: tris-(dibenzylideneacetone)dipalladium(0); potassium phosphate; tri-cyclo-hexyl-phosphine / 1,4-dioxane / 1 h / 100 °C / Microwave irradiation 2: trifluoroacetic acid / dichloromethane / 0.5 h / 20 °C View Scheme
参考文献
Choi, Jun Yong; Plummer, Mark S.; Starr, Jeremy; Desbonnet, Charlene R.; Soutter, Holly; Chang, Jeanne; Miller, J. Richard; Dillman, Keith; Miller, Alita A.; Roush, William R.
Journal of Medicinal Chemistry, 2012 , vol. 55, # 2 p. 852 - 870