1: With potassium hydrogen fluoride in methanol; water 0.5 h; 2: With chloro-trimethyl-silane; water in acetonitrile 1 h;
参考文献
O'Connell, Daniel P.; Leblanc, Daniel F.; Cromley, Debra; Billheimer, Jeffrey; Rader, Daniel J.; Bachovchin, William W.
Bioorganic and Medicinal Chemistry Letters, 2012 , vol. 22, # 3 p. 1397 - 1401