反应条件
1: formic acid; Pd2Cl2[PPh3]2; tributyl-amine; 1,3-bis-(diphenylphosphino)propane / N,N-dimethyl-formamide / 80 °C 2: palladium 10 on activated carbon; hydrogen / methanol; ethyl acetate / 20 °C 3: hydrogenchloride; water / acetonitrile / 80 °C View Scheme
参考文献
Ishii, Hideki; Koyama, Hiroko; Hagiwara, Kyoji; Miura, Tomoyuki; Xue, Guangai; Hashimoto, Yoshie; Kitahara, Genta; Aida, Yoko; Suzuki, Masaaki
Bioorganic and Medicinal Chemistry Letters, 2012 , vol. 22, # 3 p. 1469 - 1474
