反应条件
2: 1.) oxalyl chloride, 2.) pyridine / 1.) room temperature, 30 min, 2.) CH2Cl2, ice-bath, 1 h; room temperature, 2 h View Scheme
参考文献
Nakai; Konno; Kosuge; Sakuyama; Toda; Arai; Obata; Katsube; Miyamoto; Okegawa; Kawasaki
Journal of Medicinal Chemistry, 1988 , vol. 31, # 1 p. 84 - 91