反应条件
1: POCl3, Na2CO3 / 60 - 110 °C 2: 18 percent / aq. NaOH / methanol / 1.) RT, 24 h, b) 50 deg C, 3 h View Scheme
参考文献
Kukla; Breslin; Diamond; Grous; Ho; Miranda; Rodgers; Sherrill; De Clercq; Pauwels; Andries; Moens; Janssen
Journal of Medicinal Chemistry, 1991 , vol. 34, # 11 p. 3187 - 3197