反应条件
1: 95 percent / pyridine, 4-(dimethylamino)pyridine / Ambient temperature 2: 1) KF, KHCO3, 2) 30percent H2O2 / 1) THF, MeOH, 2) THF, MeOH, 60 deg C, 15 h View Scheme
参考文献
Buynak, John D.; Strickland, J. Byron; Lamb, Grady W.; Khasnis, Dipti; Modi, Seema; et al.
Journal of Organic Chemistry, 1991 , vol. 56, # 25 p. 7076 - 7083