反应条件
1: 2-methyl-1H-imidazole With sodium hydride in N,N-dimethyl-formamide; mineral oil T=20°C; 1.5 h; Inert atmosphere; 2: benzyl chloride in N,N-dimethyl-formamide; mineral oil T=0 - 50°C; Inert atmosphere;
参考文献
MacCallini, Cristina; Patruno, Antonia; Lannutti, Fabio; Ammazzalorso, Alessandra; De Filippis, Barbara; Fantacuzzi, Marialuigia; Franceschelli, Sara; Giampietro, Letizia; Masella, Simona; Felaco, Mario; Re, Nazzareno; Amoroso, Rosa
Bioorganic and Medicinal Chemistry Letters, 2010 , vol. 20, # 22 p. 6495 - 6499