反应条件
1: 82 percent / methanol / 52 h / 25 °C 2: 66.8 percent / I2, KIO3, 5 N H2SO4 / H2O; acetonitrile / 4 h / 60 °C 3: 80 percent / NaOH, water / dioxane / 1.5 h / 25 °C View Scheme
参考文献
Kumar; Knaus; Wiebe; Allen; Tempest
European Journal of Medicinal Chemistry, 1991 , vol. 26, # 5 p. 557 - 562