反应条件
1: 30percent HBr / 1) 0 deg C, 15 min, 2) rt, 4 h 2: 1) 30percent HBr, AcOH, 2) EtONa / 1) EtOH, reflux, 2) EtOH, rt View Scheme
参考文献
Schiefer, Isaac T.; Tapadar, Subhasish; Litosh, Vladislav; Siklos, Marton; Scism, Rob; Wijewickrama, Gihani T.; Chandrasena, Esala P.; Sinha, Vaishali; Tavassoli, Ehsan; Brunsteiner, Michael; Fa', Mauro; Arancio, Ottavio; Petukhov, Pavel; Thatcher, Gregory R. J.
Journal of Medicinal Chemistry, 2013 , vol. 56, # 15 p. 6054 - 6068