1N-BOC4-(2-甲基-4-硝基苯氧基)哌啶合成路线 （共 2 条）
反应条件
triphenylphosphine; diethylazodicarboxylate in dichloromethane T=20°C; Mitsunobu reaction; 18 h;
参考文献
Chemical and Pharmaceutical Bulletin, , vol. 56, # 6 p. 758 - 770
反应条件
1: 1-(tert-Butyloxycarbonyl)-4-piperidinol With sodium in DMF (N,N-dimethyl-formamide) T=5 - 15°C; 0.5 h; 2: 1-Fluoro-2-methyl-4-nitrobenzene in DMF (N,N-dimethyl-formamide) T=5 - 20°C; 3 h;
参考文献
US2004/242604 A1, ;
Page 17; 23-24 ;
US 20040242604 A1
