反应条件
1: tetrakis(triphenylphosphine) palladium(0); tri-n-butyl-tin hydride / N,N-dimethyl-formamide / 0.75 h / 100 °C / Inert atmosphere
2: methanol; copper(l) iodide / N,N-dimethyl-formamide / 5 h / 120 °C / Inert atmosphere
View Scheme
参考文献
Bhosale, Shrikar M.; Momin, Aadil A.; Kusurkar, Radhika S.
Tetrahedron, 2012 , vol. 68, # 32 p. 6420 - 6426