1: (E)-4-ethoxy-4-oxobut-2-enoic acid With pivaloyl chloride; triethylamine in tetrahydrofuran T=-10°C; 1 h; 2: oxazolidin-2-one With lithium chloride in tetrahydrofuran T=20°C; 5 h; Further stages.;
参考文献
Evans; Scheidt; Johnston; Willis
Journal of the American Chemical Society, 2001 , vol. 123, # 19 p. 4480 - 4491