甲基(1S,4R)-4-氨基-2-环戊烯-1-羧酸酯合成路线 （共 9 条）
反应条件
hydrogenchloride in various solvent(s) 24 h; Ambient temperature; Yield given;
参考文献
Tetrahedron Asymmetry, , vol. 7, # 8 p. 2381 - 2386
反应条件
1: 70 percent / aq. K2CO3 / 6 h / Ambient temperature; Irradiation 2: 43 percent / various solvent(s) / 0.5 h / Ambient temperature; immobilized lipase PS on diatomite 3: 90 percent / H2O / diisopropyl ether / 3 h / Ambient temperature; lipase PS 4: aq. HCl / 2 h / Heating 5: aq. HCl / various solvent(s) / 24 h / Ambient temperature View Scheme
参考文献
Tetrahedron Asymmetry, , vol. 7, # 8 p. 2381 - 2386
反应条件
1: 43 percent / various solvent(s) / 0.5 h / Ambient temperature; immobilized lipase PS on diatomite 2: 90 percent / H2O / diisopropyl ether / 3 h / Ambient temperature; lipase PS 3: aq. HCl / 2 h / Heating 4: aq. HCl / various solvent(s) / 24 h / Ambient temperature View Scheme
参考文献
Tetrahedron Asymmetry, , vol. 7, # 8 p. 2381 - 2386
反应条件
1: aq. HCl / 2 h / Heating 2: aq. HCl / various solvent(s) / 24 h / Ambient temperature View Scheme
参考文献
Tetrahedron Asymmetry, , vol. 7, # 8 p. 2381 - 2386
反应条件
1: 41 percent / H2O / diisopropyl ether / 3 h / Ambient temperature; lipase PS 2: aq. HCl / 2 h / Heating 3: aq. HCl / various solvent(s) / 24 h / Ambient temperature View Scheme
参考文献
Tetrahedron Asymmetry, , vol. 7, # 8 p. 2381 - 2386
反应条件
1: 90 percent / H2O / diisopropyl ether / 3 h / Ambient temperature; lipase PS 2: aq. HCl / 2 h / Heating 3: aq. HCl / various solvent(s) / 24 h / Ambient temperature View Scheme
参考文献
Tetrahedron Asymmetry, , vol. 7, # 8 p. 2381 - 2386
反应条件
hydrogenchloride 10 h; Heating;
参考文献
Journal of Medicinal Chemistry, , vol. 44, # 25 p. 4379 - 4392
反应条件
1: 2 M HCl / 72 h / Ambient temperature 2: 12 h / Heating View Scheme
参考文献
Tetrahedron Letters, , vol. 38, # 30 p. 5371 - 5374
反应条件
triethylamine in dichloromethane
1 h;
参考文献
Chand; Montgomery; Kotian; Dehghani; El-Kattan; Lin; Hutchison; Babu; Bantia; Elliott
Journal of Medicinal Chemistry, 2001 , vol. 44, # 25 p. 4379 - 4392
