反应条件
1: 1.) LiHMDS / 1.) THF, -78-0 deg C, 30 min, 2.) THF, a.) -78 deg, 30 min, b.) -78 deg C - RT, 2 h 2: NaOMe / methanol / 18 h / Heating View Scheme
参考文献
Rowley, Michael; Leeson, Paul D.; Stevenson, Graeme I.; Moseley, Angela M.; Stansfield, Ian; et al.
Journal of Medicinal Chemistry, 1993 , vol. 36, # 22 p. 3386 - 3396