5-甲基-3,4-二氨基吡啶合成路线 (共 1 条)
反应条件
hydrogenchloride; iron in ethanol 3 h; Heating / reflux;
参考文献
K.U. LEUVEN RESEARCH and DEVELOPMENT; GILEAD SCIENCES, INC.; PUERSTINGER, Gerhard
Patent: WO2005/63744 A2, 2005 ;
Location in patent: Page/Page column 232 ;