反应条件
1: 3-iodo-4-nitro-1H-pyrrolo[2,3-b]pyridine With sodium hydride in N,N-dimethyl-formamide T=0°C; 0.75 h; 2: methyl iodide in N,N-dimethyl-formamide T=0°C; 1 h;
参考文献
GLAXO WELLCOME MANUFACTURING PTE LTD; CHEN, Deborah, W.; DUNCAN, Sarah; KING, Nigel, Paul; LEE, Kiew, Ching; MAK, Sing, Yeung; RIVERS, Dean, Andrews
Patent: WO2012/170752 A1, 2012 ;
Location in patent: Page/Page column 38 ;
WO 2012/170752 A1
