1: tri-isopropoxy-borane; 1-bromo-4-fluoro-2-methylbenzene With n-butyllithium in tetrahydrofuran T=-78°C; 2: water; sodium hydroxide in tetrahydrofuran
参考文献
BIOENERGENIX; MCCALL, John M.; ROMERO, Donna L.; KELLY, Robert C.
Patent: WO2012/119046 A2, 2012 ;
Location in patent: Page/Page column 248 ;