反应条件
<b>Multi-step reaction with 3 steps<br /> </b>1: 29 percent / triphenylphosphine, iodine, pyridine / dioxane / 7 h / Ambient temperature<br />2: 78 percent / sodium methoxide / methanol / 16 h / Heating<br />3: 50 percent / imidazole / dimethylformamide / 1.25 h / Ambient temperature<br /> <br />
参考文献
Maag; Rydzewski; McRoberts; Crawford-Ruth; Verheyden; Prisbe Journal of Medicinal Chemistry, 1992 , vol. 35, # 8 p. 1440 - 1451