反应条件
1: Et3N / toluene / 3 h / Heating 2: HBr / acetic acid 3: 1.) NaH / 1.) DMF, RT, 1.5 h, 2.) DMF, RT, overnight View Scheme
参考文献
Klunder, Janice M.; Hargrave, Karl D.; West, MaryAnn; Cullen, Ernest; Pal, Kollol; et al.
Journal of Medicinal Chemistry, 1992 , vol. 35, # 10 p. 1887 - 1897