1: 4-(dihydroxyboryl)benzoic acid With N,N-diethanolaminomethyl polystyrene in tetrahydrofuran T=20°C; 1 h; 2: aniline With water; benzotriazol-1-ol; diisopropyl-carbodiimide T=20°C; 18 h; 3: in tetrahydrofuran; water T=20°C; 0.0166667 h; Further stages.;
参考文献
Gravel, Michael; Thompson, Kim A.; Zak, Mark; Berube, Christian; Hall, Dennis G.
Journal of Organic Chemistry, 2002 , vol. 67, # 1 p. 3 - 15
1: 4-(dihydroxyboryl)benzoic acid With benzotriazol-1-ol; O-(1H-benzotriazol-1-yl)-N,N,N',N'-tetramethyluronium hexafluorophosphate; N-ethyl-N,N-diisopropylamine in N,N-dimethyl-formamide 2: (cyclopropylmethyl)amine in N,N-dimethyl-formamide Further stages.;
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 18, # 1 p. 324 - 328
1: With tetrakis(triphenylphosphine) palladium(0); potassium carbonate in ethanol; water; toluene Suzuki coupling; 48 h; Inert atmosphereReflux; 2: With hydrogenchloride in water pH=3;
参考文献
Venkatraj, Muthusamy; Messagie, Jonas; Joossens, Jurgen; Lambeir, Anne-Marie; Haemers, Achiel; Van Der Veken, Pieter; Augustyns, Koen
Bioorganic and Medicinal Chemistry, 2012 , vol. 20, # 4 p. 1557 - 1568
