1: 3-methoxy-4-hydroxybenzylamine hydrochloride With sodium hydrogencarbonate in water
T=20°C; 0.5 h;
2: butyryl chloride in chloroform; water
T=20°C; 0.5 h;
in diethyl ether; N,N-dimethyl-formamide
Ambient temperature;
参考文献
Janusz, John M.; Buckwalter, Brian L.; Young, Patricia A.; LaHann, Thomas R.; Farmer, Ralph W.; et al.
Journal of Medicinal Chemistry, 1993 , vol. 36, # 18 p. 2595 - 2604
