5-溴-2-(4-甲基哌嗪-1-基)嘧啶合成路线 (共 1 条)
反应条件
1: With potassium acetate in 1,4-dioxane 0.25 h; 2: With tri-cyclo-hexyl-phosphine; tris-(dibenzylideneacetone)dipalladium(0) in 1,4-dioxane T=80°C; 2.25 h;
参考文献
PROLYSIS LTD
Patent: WO2009/74812 A1, 2009 ;
Location in patent: Page/Page column 68 ;
WO 2009/074812 A1