反应条件
1: lithium aluminium tetrahydride; AlCl3, aluminium chloride / tetrahydrofuran / 2.5 h / 1 - 10 °C
2: palladium on activated charcoal; ammonium formate / ethanol; water / 4.5 h / 50 °C / |Inert atmosphere
View Scheme
参考文献
ASTRAZENECA AB; ASTRAZENECA UK LIMITED; JOHANSSON, Lars, Anders, Mikael
Patent: WO2013/11285 A1, 2013 ;
WO 2013/011285 A1