反应条件
1: 99 percent / bis(triphenylphosphine)palladium dichloride, CuI, Et3N / dimethylformamide / 2 h / 70 °C 2: 80 percent / NH3 / methanol / 3 h / 80 °C 3: 96 percent / 80percent aq. TFA / 2 h / Ambient temperature View Scheme
参考文献
Homma, Hiroshi; Watanabe, Yohko; Abiru, Toichi; Murayama, Toshihiko; Nomura, Yasuharu; Matsuda, Akira
Journal of Medicinal Chemistry, 1992 , vol. 35, # 15 p. 2881 - 2890
