1-(4-硝基苯基)-1H-四唑合成路线 （共 14 条）
反应条件
acetic acid T=100°C; 0.166667 h;
参考文献
Karimi Zarchi, Mohammad Ali; Nazem, Fatemeh
Journal of the Iranian Chemical Society, 2014 , vol. 11, # 1 p. 91 - 99
反应条件
potassium carbonate in N,N-dimethyl-formamide T=80°C;
参考文献
MERCK CANADA INC.; BOYD, Michael John; CHIASSON, Jean-François; CRANE, Sheldon; GIROUX, André
Patent: WO2013/59928 A1, 2013 ;
Location in patent: Page/Page column 33 ;
反应条件
hydrogenchloride; methanol; trimethylsilylazide in diethyl ether T=60°C; 4 h;
参考文献
Jin, Tienan; Kamijo, Shin; Yamamoto, Yoshinori
Tetrahedron Letters, 2004 , vol. 45, # 51 p. 9435 - 9437
反应条件
trimethylsilylazide; triphenylphosphine; diethylazodicarboxylate in tetrahydrofuran 24 h;
参考文献
Bristol-Myers Squibb Pharma Company
Patent: EP946508 B1, 2009 ;
Location in patent: Page/Page column 68 ;
反应条件
trimethylsilylacetylene; zinc(II) chloride in chloroform 20 h; Heating;
参考文献
Nishiyama, Kozaburo; Oba, Makoto; Watanabe, Akio
Tetrahedron, 1987 , vol. 43, # 4 p. 693 - 700
反应条件
sodium azide; acetic acid T=83°C; 2 h;
参考文献
Ichikawa, Takashi; Kitazaki, Tomoyuki; Matsushita, Yoshihiro; Hosono, Hiroshi; Yamada, Masami; Mizuno, Masahiro; Itoh, Katsumi
Chemical and Pharmaceutical Bulletin, 2000 , vol. 48, # 12 p. 1947 - 1953
参考文献
Freund; Paradies
Chemische Berichte, 1901 , vol. 34, p. 3120
参考文献
Dimroth; de Montmollin
Chemische Berichte, 1910 , vol. 43, p. 2914
反应条件
methanol; diethyl ether
参考文献
Huisgen; Koch
Justus Liebigs Annalen der Chemie, 1955 , vol. 591, p. 200,221
参考文献
Huisgen; Koch
Justus Liebigs Annalen der Chemie, 1955 , vol. 591, p. 200,221
