1: 93.2 percent / Et3N / acetic acid / 6 h / Ambient temperature
2: 87.3 percent / NH3 / ethanol / Ambient temperature
View Scheme
参考文献
Bannyi, I. P.; Chernykh, V. P.; Petyunin, P. A.; Chuvurin, A. V.; Chaleeva, L. D.; et al.
Pharmaceutical Chemistry Journal, 1982 , vol. 16, # 1 p. 33 - 37
Khimiko-Farmatsevticheskii Zhurnal, 1982 , vol. 16, # 1 p. 43 - 47
1: 93.2 percent / Et3N / acetic acid / 6 h / Ambient temperature
2: 67.1 percent / ethanol / Ambient temperature
View Scheme
参考文献
Bannyi, I. P.; Chernykh, V. P.; Petyunin, P. A.; Chuvurin, A. V.; Chaleeva, L. D.; et al.
Pharmaceutical Chemistry Journal, 1982 , vol. 16, # 1 p. 33 - 37
Khimiko-Farmatsevticheskii Zhurnal, 1982 , vol. 16, # 1 p. 43 - 47