2-氯-4-氨基-5-[(三甲基硅基)乙炔基]苯腈合成路线 (共 1 条)
反应条件
1: tetrabutyl ammonium fluoride / tetrahydrofuran / 75 °C 2: potassium sec-butoxide / tetrahydrofuran / 3 h / 75 °C View Scheme
参考文献
F. HOFFMANN-LA ROCHE AG; ALIAGAS-MARTIN, Ignacio; CRAWFORD, James; LEE, Wendy; MATHIEU, Simon; RUDOLPH, Joachim
Patent: WO2013/26914 A1, 2013 ;
WO 2013/026914 A1