1: With dimethylsulfide borane complex in tetrahydrofuran T=0°C; 19 h; Reflux; 2: With methanol 18 h; Reflux;
参考文献
BRISTOL-MYERS SQUIBB COMPANY; ORWAT, Michael J.; PINTO, Donald J.P.; SMITH II, Leon M.; SRIVASTAVA, Shefali
Patent: WO2013/56034 A1, 2013 ;
Location in patent: Paragraph 003606 ;