1: benzyl-methyl-amine With sodium hydride in tetrahydrofuran T=0°C; 0.25 h; 2: (R/S)-2-Bromomethyl-oxirane in tetrahydrofuran Heating; Further stages.;
参考文献
Robin, Aelig; Brown, Fraser; Bahamontes-Rosa, Noemi; Wu, Binghua; Beitz, Eric; Kun, Juergen F. J.; Flitsch, Sabine L.
Journal of Medicinal Chemistry, 2007 , vol. 50, # 17 p. 4243 - 4249