反应条件
1: 83 percent / Et3N / CH2Cl2 / 0.5 h / 0 °C 2: 76 percent / glacial acetic acid, NaI, KI / H2O / 1 h / Heating 3: 1.) NaBH4, 2.) HCHO, HCl / 1.) ethanol, r.t., 2 h; 2.) water, 80 deg C, 10 min View Scheme
参考文献
Acta Chimica Hungarica, , vol. 124, # 2 p. 209 - 216