反应条件
<b>Multi-step reaction with 3 steps<br /> </b>1: 1) NaH, n-BuLi / 1) THF, -20 deg C<br />2: NaBH<sub>4</sub>, BEt<sub>3</sub> / tetrahydrofuran; methanol / -78 °C<br />3: H+<br /> <br />
参考文献
Balasubramanian, N.; Brown, P. J.; Catt, J. D.; Han, W. T.; Parker, R. A.; et al. Journal of Medicinal Chemistry, 1989 , vol. 32, # 9 p. 2038 - 2041