反应条件
1: N,N-dimethyl-3-(thien-2-yl)-3-hydroxy-propanamine With sodium hydride in dimethyl sulfoxide T=20°C; 2: 4-fluoro-l-naphthalene in dimethyl sulfoxide T=48 - 50°C; 3: oxalic acid in ethyl acetate T=20°C; 5 h;
参考文献
JUBILANT LIFE SCIENCES LIMITED; BISWAS, Sujay; TRIVEDI, Archana; KHARBANDA, Manlta; DUBEY, Shailendra; SINGLA, Sandeep; YOGIRAJ, Mansukhlal, Bodheka; VIR, Dharam
Patent: WO2011/33366 A2, 2011 ;
Location in patent: Page/Page column 23 ;