1-叔丁氧羰基-4-氨甲基哌啶合成路线 （共 27 条）
反应条件
1: toluene / Heating 2: toluene / 25 °C 3: aq. KHSO4 View Scheme
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 16, # 19 p. 5212 - 5216
反应条件
in methanol T=-30 - 23°C; 16 h;
参考文献
EP1032561 B1, ;
Page 10 ;
EP 1032561 B1
反应条件
p-toluenesulfonic acid monohydrate; triethylamine in N,N-dimethyl-formamide
参考文献
US2003/119811 A1, ;
US 20030119811 A1
反应条件
1.1: ClCOO-i-Bu; N-methylmorpholine 1.2: aq. NH3 2.1: LiAlH4 View Scheme
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 12, # 5 p. 757 - 761
反应条件
1: Et3N / CH2Cl2 / 0 °C 2: NaN3 / dimethylformamide / Heating 3: 100 percent / H2 / 10 percent Pd/C / methanol View Scheme
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 11, # 24 p. 3161 - 3164
反应条件
1: NaN3 / dimethylformamide / Heating 2: 100 percent / H2 / 10 percent Pd/C / methanol View Scheme
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 11, # 24 p. 3161 - 3164
反应条件
1: 100 percent / CH2Cl2 2: 100 percent / BH3*THF / tetrahydrofuran 3: Et3N / CH2Cl2 / 0 °C 4: NaN3 / dimethylformamide / Heating 5: 100 percent / H2 / 10 percent Pd/C / methanol View Scheme
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 11, # 24 p. 3161 - 3164
反应条件
1: toluene / 25 °C 2: aq. KHSO4 View Scheme
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 16, # 19 p. 5212 - 5216
反应条件
1: 59 percent / TEA / CH2Cl2 2: 100 percent / NH2NH2*H2O / ethanol View Scheme
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 11, # 10 p. 1261 - 1264
